Valemetostat (DS-3201)

InformationValemetostat (DS-3201) Valemetostat (DS-3201, DS-3201b) is a selective EZH1/2 dual inhibitor.TargetsEZH1 ; EZH2In vitroValemetostat significantly reducs ATL cell viability compared with the others. Valemetostat significantly reactivates the expression of the highly H3K27me3-accumulated EZH1/2 target genes in an ex vivo culture of primary ATL cells. Valemetostat shows superior anti-growth effects compared with EZH2-selective inhibitor in malignant lymphoma cell lines..Cell Research(from reference)Cell lines：23 cell lines derived from hematological malignancies Incubation Time：1, 7, 14 days

Specifictaions: Moligand™, ≥98%

MDL Number: C26H34ClN3O4 

Molecular Formula: 488.02

PubChem CID: 126481870

Isomeric SMILES: CC1=CC(=C(C(=O)N1)CNC(=O)C2=CC(=C3C(=C2C)O[C@@](O3)(C)C4CCC(CC4)N(C)C)Cl)C

UPC:

51291603

Condition:

New

Weight:

1.06 Ounces

HazmatClass:

No

Quantity:

1

Unit of Measurement:

EA

WeightUOM:

LB

MPN:

V414273-1mg

CAS:

1809336-39-7

Product Size:

1mg